Description

Cabergoline (Dostinex) Description

Cabergoline (Dostinex) is a selective dopamine receptor agonist. This agent is highly specific in its actions, with a strong affinity for the dopamine D2 receptor, and a low affinity for serotonin, and 5-HT2-serotonin receptors. Its main clinical use is for the treatment of hyperprolactinemia, or the hyper-secretion of prolactin from lactotrophs in the anterior pituitary (pituitary tumor is a common cause of this disorder). It is also applied in the management of Parkinson’s disease. Cabergoline effectively inhibits prolactin secretion, which it does by mimicking the actions of dopamine on the D2 receptor (dopamine normally serves as negative feedback for prolactin release). As a targeted agonist of the dopamine D2 receptor, cabergoline should not affect other pituitary hormones like growth hormone (GH), luteinizing hormone (LH), corticotrophin (ACTH), or thyroid-stimulating hormone (TSH).

Cabergoline works directly to inhibit prolactin secretion in the pituitary gland’s lactotroph cells. In actuality, the function of the drug is incredibly simple, and that’s why it’s so interesting to a lot of people.

This ensures that one can maximize the most out of Cabergoline, even if you’re not planning to be a world champion athlete. In fact, some of the users use it in personal life are for sexual performance. For the athlete, however, the primary reason they would need caber is due to their use of Anabolics.

Athletes like Cabergoline because they enjoy the rush that often comes from increased dopamine.

Positive Effects of Cabergoline (Dostinex)

Positives of using Cabergoline is the positive sleep effects that people report on it. For many Caber users, they claim they get deeper, more restful sleep. And lastly, they also report that there is a tremendous increase in sex drive.

Dosages

Dosages are falling in the range of 0.25 mg up to 1 mg twice per week, from 0.5 mg up to 2 mg per week.